SCHEMBL8300934

SCHEMBL8300934

N=C(Nc1ccccc1OC(F)(F)F)N1CCCc2cc(C(F)(F)F)ccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.41
GAA P10253 2/20 0.41
HTR2A P28223 3/20 0.40
HTR2C P28335 3/20 0.40
HTR2B P41595 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 3/20 0.38
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
GPBAR1 Q8TDU6 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
P2RY1 P47900 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8334504 0.87 GAA (0.54) NOTUMGAAMEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL6775779 0.86 GAA (0.53) NOTUMGAAMEN1KMT2ALMNA
SCHEMBL7106084 0.76 NOTUM (0.41) NOTUMHTR2AHTR2CHTR2BMEN1
SCHEMBL8332662 0.73 MAPT (0.42) NOTUMHTR2AHTR2CLMNACYP3A4
SCHEMBL8522982 0.72 ALDH1A1 (0.41) NOTUMHTR2AHTR2CMEN1KMT2A
SCHEMBL8524737 0.72 MAPT (0.43) NOTUMHTR2AHTR2CMEN1KMT2A
SCHEMBL8331768 0.72 ALDH1A1 (0.57) HTR2CMEN1KMT2ALMNAP2RY1
SCHEMBL8334232 0.69 XPO1 (0.39) NOTUMHTR2AHTR2CMEN1KMT2A
SCHEMBL7552151 0.69 NOTUM (0.63) NOTUMHTR2AHTR2CMEN1KMT2A
Hydrochloric Acid SCHEMBL6774819 0.68 XPO1 (0.39) NOTUMHTR2AHTR2CMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0925300-A4 1999-06-30 EP claimed
EP-0925300-A1 PHARMACEUTICALLY ACTIVE COMPOUNDS AND METHODS OF USE CAMBRIDGE NEUROSCIENCE, INC. (US) 1999-06-30 EP claimed
WO-1997030054-A1 PHARMACEUTICALLY ACTIVE COMPOUNDS AND METHODS OF USE CAMBRIDGE NEUROSCIENCE, INC. (US) 1997-08-21 WO claimed