SCHEMBL8334232

SCHEMBL8334232

N=C(Nc1cc(Br)ccc1Br)N1CCCc2ccc(C(F)(F)F)cc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XPO1 O14980 2/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
CNR2 P34972 1/20 0.38
CCKBR P32239 1/20 0.36
CPT2 P23786 1/20 0.35
CPT1A P50416 1/20 0.35
CPT1B Q92523 1/20 0.35
HDAC1 Q13547 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
FGFR4 P22455 1/20 0.34
ERAP1 Q9NZ08 1/20 0.34
P2RX1 P51575 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6774819 0.99 XPO1 (0.39) XPO1HTR2AHTR2CCNR2CCKBR
SCHEMBL8332799 0.75 ALDH1A1 (0.40) HTR2AHTR2CCNR2ALDH1A1MAPT
SCHEMBL8337181 0.75 ALDH1A1 (0.40) HTR2AHTR2CCNR2P2RX1MEN1
SCHEMBL6775028 0.75 SIGMAR1 (0.50) MEN1KMT2AALDH1A1MAPTNOTUM
Hydrochloric Acid SCHEMBL6769802 0.74 ALDH1A1 (0.41) HTR2AHTR2CHDAC1HDAC6HDAC3
Hydrochloric Acid SCHEMBL6774822 0.74 CNR2 (0.37) XPO1HTR2AHTR2CCNR2CPT2
SCHEMBL7743748 0.73 ALDH1A1 (0.39) HTR2AHTR2CCNR2FGFR4ERAP1
SCHEMBL331761 0.72 PDK1 (0.52) HTR2AHTR2CCNR2MEN1KMT2A
SCHEMBL27544652 0.70 CNR2 (0.53) HTR2AHTR2CCNR2CPT2CPT1A
SCHEMBL10241674 0.69 NOTUM (0.66) HTR2AHTR2CCNR2XIAPBIRC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999002145-A1 COMBINATION DRUG THERAPIES COMPRISING AMINOGLYCOSIDE ANTIBIOTICS AND N,N'-DISUBSTITUTED GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1999-01-21 WO disclosed