SCHEMBL8301017

SCHEMBL8301017

CCOC(=O)C(CCc1ccccc1)NCCCCCN

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR2 O60603 2/20 0.51
CHRNB2 P17787 1/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CHRNA4 P43681 1/20 0.49
ACE P12821 5/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
GGT1 P19440 1/20 0.44
HPRT1 P00492 1/20 0.44
MMP8 P22894 1/20 0.44
ABCB11 O95342 2/20 0.44
SIRT2 Q8IXJ6 1/20 0.43
SIRT1 Q96EB6 1/20 0.43
SIRT3 Q9NTG7 1/20 0.43
LMNA P02545 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273868 0.85 SMN1; SMN2 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4ACE
SCHEMBL8302557 0.83 TLR2 (0.41) TLR2CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL27458051 0.81 ACE (0.58) TLR2ACESMN1; SMN2ABCB11LMNA
SCHEMBL6237696 0.81 ACE (0.58) TLR2ACESMN1; SMN2ABCB11LMNA
SCHEMBL6240311 0.81 ACE (0.58) TLR2ACESMN1; SMN2ABCB11LMNA
Hydrochloric Acid SCHEMBL11206033 0.81 SMN1; SMN2 (0.50) ACESMN1; SMN2MMP8ABCB11LMNA
Bromide SCHEMBL11083780 0.80 ALOX5 (0.49) GGT1SIRT2SIRT1
SCHEMBL14265369 0.80 SMN1; SMN2 (0.55) ACESMN1; SMN2MMP8ABCB11LMNA
SCHEMBL10482405 0.80 SMN1; SMN2 (0.55) ACESMN1; SMN2MMP8ABCB11LMNA
Water SCHEMBL28202314 0.80 TLR2 (0.59) TLR2SIRT2SIRT1SIRT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1635816-B1 ENALAPRIL-NITROXYDERIVATIVES DERIVATIVES AND RELATED COMPOUNDS AS ACE INHIBITORS FOR THE TREATMENT OF CARDIOVASCULAR DISEASES NICOX SA (FR) 2009-03-04 EP disclosed
WO-2004110432-A1 ENALAPRIL-NITROXYDERIVATIVES DERIVATIVES AND RELATED COMPOUNDS AS ACE INHIBITORS FOR THE TREATMENT OF CARDIOVASCULAR DISEASES NICOX S.A. (FR) 2004-12-23 WO disclosed