SCHEMBL8301690

SCHEMBL8301690

CC(C)(C)NC(=O)NC(C=O)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
POLB P06746 1/20 0.36
EPHX2 P34913 1/20 0.35
EPHX1 P07099 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
CTSK P43235 2/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL861760 1.00 TRPA1 (0.38) TRPA1POLBEPHX2EPHX1MEN1
SCHEMBL2019181 0.76 CTSK (0.33) CTSK
SCHEMBL13051375 0.76 CTSK (0.33) EPHX1ALOX15CTSK
SCHEMBL24441870 0.75 CYP2C9 (0.42) MEN1KMT2ACTSK
SCHEMBL14612334 0.74 CTSK (0.32) CTSK
SCHEMBL15338780 0.73 CTSK (0.33) MEN1KMT2ARAB9ACTSK
SCHEMBL7945239 0.72 CTSK (0.38) CTSK
SCHEMBL23917859 0.72 CTSK (0.32) CTSK
SCHEMBL24567754 0.71 POLB (0.45) TRPA1POLBEPHX2EPHX1MEN1
SCHEMBL18793674 0.71 POLB (0.45) TRPA1POLBEPHX2EPHX1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004113294-A1 PROCESS AND INTERMEDIATES FOR THE PREPARATION OF (1R, 2S, 5S)-3-AZABICYCLO[3, 1, 0]HEXANE-2-CARBOXAMIDE, N-[3-AMINO-1-(CYCLOBUTYLMETHYL)-2, 3-DIOXOPROPYL] ]-3-[(2S)-2-[[[1, 1-DIMETHYLETHYL]AMINO]CARBONYLAMINO]-3, 3-DIMETHYL-1-OXOBUTYL]-6, 6-DIMETHYL SCHERING CORPORATION (US) 2004-12-29 WO disclosed