SCHEMBL8301971

SCHEMBL8301971

O=C1CCCc2cc(C(O)CN3CCC(CCC4CCCCC4)CC3)ccc2N1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.52
GRIN2B Q13224 2/20 0.48
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
ALDH1A1 P00352 3/20 0.42
ATM Q13315 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
GSK3B P49841 1/20 0.38
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
OGT O15294 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8439768 0.91 KCNH2 (0.54) KCNH2GRIN2BHTR1ADRD2HTR2A
SCHEMBL8301786 0.90 HTR1A (0.53) KCNH2GRIN2BHTR1ADRD2HTR2A
Hydrochloric Acid SCHEMBL8542941 0.84 MEN1 (0.56) KCNH2GRIN2BALDH1A1ATMLMNA
SCHEMBL466863 0.81 GRIN2B (0.61) KCNH2GRIN2BHTR1ADRD2HTR2A
SCHEMBL9562497 0.80 KCNH2 (0.57) KCNH2GRIN2BHTR1ADRD2HTR2A
SCHEMBL9562478 0.80 GRIN2B (0.60) KCNH2GRIN2BHTR1ADRD2HTR2A
SCHEMBL9562529 0.80 KCNH2 (0.57) KCNH2GRIN2BHTR2ATSHRTP53
SCHEMBL9562489 0.80 KCNH2 (0.51) KCNH2GRIN2BHTR1ADRD2HTR2A
Hydrochloric Acid SCHEMBL8548193 0.80 GRIN2B (0.55) KCNH2GRIN2BALDH1A1ATMOGT
Hydrochloric Acid SCHEMBL8548360 0.80 GRIN2B (0.55) KCNH2GRIN2BALDH1A1ATMOGT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848707-B1 4-(CYCLOALKYL)PIPERIDINES AND 4-(CYCLOALKYLALKYL)-PIPERIDINES DERIVATIVES, PREPARATION THEREOF AND THERAPEUTICAL APPLICATIONS THEREOF SYNTHELABO (FR) 1999-08-04 EP disclosed