SCHEMBL8303972

SCHEMBL8303972

CC1CCN(S(=O)(=O)c2ccc3[nH]c(=O)cc(C(=O)NCc4ccccn4)c3c2)CC1

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.64
HTT P42858 2/20 0.63
KDM4E B2RXH2 1/20 0.63
NPC1 O15118 1/20 0.57
TDP1 Q9NUW8 2/20 0.56
TP53 P04637 1/20 0.56
KMT2A Q03164 3/20 0.55
ALDH1A1 P00352 2/20 0.55
MEN1 O00255 2/20 0.55
USP2 O75604 2/20 0.55
HSP90AA1 P07900 1/20 0.55
HSP90AB1 P08238 1/20 0.55
HPGD P15428 1/20 0.55
YWHAG P61981 1/20 0.55
RXFP1 Q9HBX9 2/20 0.53
LMNA P02545 2/20 0.53
MAPT P10636 2/20 0.53
GAA P10253 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312226 0.90 TDP1 (0.67) BACE1HTTKDM4ENPC1TDP1
SCHEMBL8311500 0.90 TDP1 (0.67) BACE1HTTKDM4ENPC1TDP1
SCHEMBL8305689 0.85 LMNA (0.69) BACE1HTTKDM4ETDP1TP53
SCHEMBL8304644 0.85 LMNA (0.66) BACE1HTTKDM4ETDP1TP53
SCHEMBL8304348 0.83 BACE1 (0.68) BACE1HTTKDM4ETDP1TP53
SCHEMBL8304646 0.80 KDM4E (0.76) BACE1HTTKDM4ENPC1TP53
SCHEMBL8308406 0.79 KDM4E (0.74) BACE1HTTKDM4ENPC1TP53
SCHEMBL8308301 0.79 KDM4E (0.74) BACE1HTTKDM4ETDP1TP53
SCHEMBL8308894 0.78 KDM4E (0.70) BACE1HTTKDM4ETP53KMT2A
SCHEMBL8308219 0.78 KDM4E (0.72) BACE1HTTKDM4ETP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed