SCHEMBL8312226

SCHEMBL8312226

O=C(NCc1ccccn1)c1cc(=O)[nH]c2ccc(S(=O)(=O)N3CCCCC3)cc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.67
TP53 P04637 1/20 0.66
NPC1 O15118 1/20 0.66
ALDH1A1 P00352 3/20 0.65
USP2 O75604 2/20 0.65
MEN1 O00255 1/20 0.65
HSP90AA1 P07900 1/20 0.65
HSP90AB1 P08238 1/20 0.65
HPGD P15428 1/20 0.65
YWHAG P61981 1/20 0.65
KMT2A Q03164 1/20 0.65
MAPT P10636 1/20 0.62
LMNA P02545 2/20 0.60
HTT P42858 1/20 0.60
RXFP1 Q9HBX9 1/20 0.60
BACE1 P56817 3/20 0.59
SMN1; SMN2 Q16637 1/20 0.55
KDM4E B2RXH2 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.52
TSHR P16473 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311500 1.00 TDP1 (0.67) TDP1TP53NPC1ALDH1A1USP2
SCHEMBL8303972 0.90 BACE1 (0.64) TDP1TP53NPC1ALDH1A1USP2
SCHEMBL8311835 0.86 TP53 (0.76) TDP1TP53ALDH1A1MEN1KMT2A
SCHEMBL8311212 0.86 TP53 (0.76) TDP1TP53ALDH1A1MEN1KMT2A
SCHEMBL8308783 0.85 TP53 (0.75) TDP1TP53ALDH1A1MEN1KMT2A
SCHEMBL8311830 0.84 MAPT (0.68) TDP1TP53ALDH1A1MAPTLMNA
SCHEMBL8312633 0.83 ALDH1A1 (0.69) TDP1TP53ALDH1A1USP2KMT2A
SCHEMBL8312641 0.83 TP53 (0.68) TDP1TP53ALDH1A1MAPTLMNA
SCHEMBL8308161 0.83 LMNA (0.68) TDP1TP53ALDH1A1MAPTLMNA
SCHEMBL8305995 0.82 TP53 (0.66) TDP1TP53ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed