SCHEMBL5776476

SCHEMBL5776476

CC(C)c1csc(C=Cc2cccc([N+](=O)[O-])c2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 3/20 0.52
CYP19A1 P11511 1/20 0.51
MAPT P10636 4/20 0.48
ALDH1A1 P00352 3/20 0.48
RAB9A P51151 3/20 0.48
NPC1 O15118 2/20 0.48
FBP1 P09467 1/20 0.48
VCP P55072 1/20 0.48
ALB P02768 1/20 0.48
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
LMNA P02545 2/20 0.46
HTT P42858 2/20 0.46
MCL1 Q07820 1/20 0.46
PTK2B Q14289 1/20 0.46
POLB P06746 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TRPV1 Q8NER1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9515918 1.00 NFE2L2 (0.52) NFE2L2CYP19A1MAPTALDH1A1RAB9A
SCHEMBL5778781 0.84 ALB (0.55) MAPTRAB9ANPC1ALBMEN1
SCHEMBL8304425 0.81 ALB (0.52) MAPTALDH1A1ALBMEN1KMT2A
SCHEMBL8304428 0.81 ALB (0.52) MAPTALDH1A1ALBMEN1KMT2A
SCHEMBL9268700 0.80 MAPT (0.43) MAPTALDH1A1MEN1KMT2ALMNA
SCHEMBL9256181 0.80 ALDH1A1 (0.40) MAPTALDH1A1ALBMEN1KMT2A
SCHEMBL9256170 0.80 ALDH1A1 (0.40) MAPTALDH1A1ALBMEN1KMT2A
SCHEMBL9260315 0.78 ALB (0.49) CYP19A1MAPTNPC1ALBMAOB
SCHEMBL5775275 0.78 ALB (0.52) NPC1FBP1ALBMEN1KMT2A
SCHEMBL5777449 0.78 ALB (0.49) CYP19A1MAPTNPC1ALBMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed
EP-0219436-B1 Thiazole derivative and leukotriene antagonist containing the same as the effective ingredients MITSUBISHI CHEM IND (JP) 1993-12-22 EP disclosed
US-4902700-A Thiazole derivative and leukotriene antagonist containing the same as the effective ingredients MITSUBISHI KASEI CORPORATION (JP) 1990-02-20 US disclosed
EP-0219436-A2 Thiazole derivative and leukotriene antagonist containing the same as the effective ingredients MITSUBISHI KASEI CORPORATION (JP) 1987-04-22 EP disclosed