SCHEMBL8304724

SCHEMBL8304724

C=CCc1c(N2CCNC2=N)ccc2c1NC(=O)CO2

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.34
DRD3 P35462 5/20 0.34
DRD4 P21917 5/20 0.34
NR3C2 P08235 2/20 0.31
DRD1 P21728 1/20 0.31
HTR2A P28223 1/20 0.31
PARP1 P09874 1/20 0.30
CCR1 P32246 1/20 0.30
KCNH2 Q12809 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301738 0.87 PARP1 (0.39) DRD2DRD3DRD4NR3C2DRD1
SCHEMBL8308384 0.85 DRD2 (0.37) DRD2DRD3DRD4NR3C2DRD1
SCHEMBL8304731 0.82
SCHEMBL8308168 0.81 DRD2 (0.37) DRD2DRD3DRD4NR3C2HTR2A
SCHEMBL8305470 0.81 NR3C2 (0.44) DRD2DRD3DRD4NR3C2HTR2A
SCHEMBL8301771 0.76 NR3C2 (0.37) NR3C2PARP1CCR1KCNH2CYP3A4
SCHEMBL8301805 0.76 PARP1 (0.35) DRD2DRD3DRD4NR3C2PARP1
SCHEMBL8304614 0.76 PARP1 (0.35) DRD2DRD3DRD4NR3C2HTR2A
SCHEMBL8307023 0.71 DRD2 (0.38) DRD2DRD3DRD4NR3C2DRD1
SCHEMBL8303552 0.70 DRD2 (0.33) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0548254-B1 6- OR 7-(IMIDAZOLIDIN-2-YLIDENEAMINO)-1,4-BENZOXAZINES AS ALPHA ADRENERGIC AGENTS ALLERGAN INC (US) 1999-06-02 EP disclosed
US-5091528-A Antiglaucoma, antidiarrhea agents, diuretics, vasoconstrictors ALLERGAN, INC. (US) 1992-02-25 US disclosed