SCHEMBL8304925

SCHEMBL8304925

c1ccc2c(NC3NCCN3)n[nH]c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.51
TRPA1 O75762 1/20 0.47
FADS1 O60427 2/20 0.44
KDM4E B2RXH2 2/20 0.44
GAA P10253 2/20 0.44
PDPK1 O15530 1/20 0.44
CYP3A4 P08684 1/20 0.44
ACHE P22303 1/20 0.42
MAPK10 P53779 8/20 0.42
ALDH1A1 P00352 1/20 0.42
ALPL P05186 1/20 0.42
IDO1 P14902 1/20 0.42
HPGD P15428 1/20 0.42
TTK P33981 1/20 0.42
MCHR1 Q99705 1/20 0.41
MAPK8 P45983 5/20 0.40
MAPK9 P45984 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
GRM4 Q14833 1/20 0.40
AURKA O14965 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15392392 0.76 TRPA1 (0.54) ADRA2ATRPA1FADS1KDM4EGAA
SCHEMBL19100299 0.72 MAPK1 (0.49) ADRA2ATRPA1ACHEMAPK10MCHR1
SCHEMBL11700794 0.72 KDM4E (0.57) ADRA2ATRPA1FADS1KDM4EGAA
SCHEMBL11756891 0.72 TRPA1 (0.54) ADRA2ATRPA1FADS1KDM4EGAA
SCHEMBL7172053 0.72 TRPA1 (0.54) ADRA2ATRPA1FADS1KDM4EGAA
SCHEMBL7452500 0.72 TRPA1 (0.54) ADRA2ATRPA1FADS1KDM4EGAA
SCHEMBL31032755 0.72 TRPA1 (0.54) ADRA2ATRPA1FADS1KDM4EGAA
SCHEMBL2854739 0.71 TRPA1 (0.50) ADRA2ATRPA1FADS1KDM4EGAA
SCHEMBL966349 0.71 TRPA1 (0.50) ADRA2ATRPA1FADS1KDM4EGAA
SCHEMBL20812420 0.69 DDB1 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944620-A1 2-IMIDAZOLINYLAMINOINDAZOLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1999-09-29 EP disclosed
WO-1998023609-A1 2-IMIDAZOLINYLAMINOINDAZOLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1998-06-04 WO disclosed