SCHEMBL8305524

SCHEMBL8305524

CCCCCCCCOc1cnc(C2CCc3cc(OCCCCCCCC)nc(F)c3C2)nc1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 3/20 0.33
HTR1B P28222 3/20 0.33
THRA P10827 2/20 0.33
THRB P10828 2/20 0.33
TAOK3 Q9H2K8 3/20 0.33
GPR84 Q9NQS5 1/20 0.32
TAOK1 Q7L7X3 2/20 0.32
HTR1A P08908 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301529 0.87 HTR1D (0.36) HTR1DHTR1BTHRATHRBTAOK3
SCHEMBL8303039 0.80 NR5A1 (0.33) TAOK3
SCHEMBL8296395 0.78 THRA (0.32) THRATHRBTAOK3GPR84
SCHEMBL8294020 0.78 THRA (0.38) THRATHRBTAOK3GPR84TAOK1
SCHEMBL5722827 0.74 HTR1D (0.33) HTR1DHTR1BTHRATHRB
SCHEMBL9292317 0.72 NR5A1 (0.43) HTR1BTHRATHRB
SCHEMBL9292320 0.72 NR5A1 (0.43) HTR1BTHRATHRB
SCHEMBL8305593 0.69 XDH (0.40) HTR1DHTR1BTHRATHRB
SCHEMBL8293940 0.69 THRA (0.35) HTR1DHTR1BTHRATHRBTAOK3
SCHEMBL8298265 0.69 THRA (0.41) THRATHRBTAOK3GPR84TAOK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824520-B1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AG (DE) 1999-10-06 EP disclosed
EP-0824520-A1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-25 EP disclosed
WO-1996035675-A1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1996-11-14 WO disclosed