SCHEMBL8301529

SCHEMBL8301529

CCCCCCCCOc1ccc(C2CCc3cc(OCCCCCCCC)nc(F)c3C2)nc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.36
HTR1B P28222 2/20 0.36
THRA P10827 2/20 0.36
THRB P10828 2/20 0.36
TAOK3 Q9H2K8 3/20 0.35
TAOK1 Q7L7X3 2/20 0.34
HPGD P15428 3/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NR5A1 Q13285 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
GPR84 Q9NQS5 1/20 0.31
PTPN1 P18031 1/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
RAB9A P51151 1/20 0.31
CNR2 P34972 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303039 0.89 NR5A1 (0.33) TAOK3NR5A1CNR2CNR1
SCHEMBL8305524 0.87 HTR1D (0.33) HTR1DHTR1BTHRATHRBTAOK3
SCHEMBL8298265 0.79 THRA (0.41) THRATHRBTAOK3TAOK1PDE3B
SCHEMBL8293940 0.79 THRA (0.35) HTR1DHTR1BTHRATHRBTAOK3
SCHEMBL8305593 0.71 XDH (0.40) HTR1DHTR1BTHRATHRBHPGD
SCHEMBL8294020 0.69 THRA (0.38) THRATHRBTAOK3TAOK1PDE3B
SCHEMBL8296395 0.69 THRA (0.32) THRATHRBTAOK3PDE3BPDE3A
SCHEMBL8301428 0.69 THRA (0.34) THRATHRBTAOK3NR5A1GPR84
SCHEMBL8299252 0.69 NR5A1 (0.32) NR5A1GPR84CNR2CNR1
SCHEMBL10875327 0.68 NR5A1 (0.41) HTR1BTHRATHRBHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824520-B1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AG (DE) 1999-10-06 EP disclosed
EP-0824520-A1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-25 EP disclosed
WO-1996035675-A1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1996-11-14 WO disclosed