SCHEMBL8305596

SCHEMBL8305596

N=C(N)NCCC[C@H](N)C(=O)c1nc2ccccc2s1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.44
TP53 P04637 1/20 0.44
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
CASP1 P29466 1/20 0.43
ALDH1A1 P00352 1/20 0.43
ALOX5 P09917 1/20 0.43
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
PKM P14618 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
HPGD P15428 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5047017 1.00 L3MBTL1 (0.44) L3MBTL1TP53ALOX15TSHRCASP1
SCHEMBL29732021 1.00 L3MBTL1 (0.44) L3MBTL1TP53ALOX15TSHRCASP1
SCHEMBL14524820 0.88 ALOX15 (0.44) L3MBTL1TP53ALOX15TSHRCASP1
SCHEMBL14524842 0.88 ALOX15 (0.44) L3MBTL1TP53ALOX15TSHRCASP1
SCHEMBL22850476 0.88 L3MBTL1 (0.44) L3MBTL1TP53ALOX15TSHRCASP1
SCHEMBL22930256 0.86 NPC1 (0.51) L3MBTL1TP53ALOX15TSHRCASP1
SCHEMBL22930269 0.86 L3MBTL1 (0.41) L3MBTL1TP53ALOX15TSHRCASP1
SCHEMBL8667159 0.86 TP53 (0.42) L3MBTL1TP53ALOX5
SCHEMBL14127426 0.85 PRSS1 (0.48)
SCHEMBL17145027 0.84 NFKB1 (0.41) TP53ALDH1A1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7205384-B2 Process for preparing peptidyl heterocyclic ketone derivatives ORTHO-MCNEIL PHARMACEUTICAL INC. (US) 2007-04-17 US disclosed
US-7205384-B2 Process for preparing peptidyl heterocyclic ketone derivatives ORTHO-MCNEIL PHARMACEUTICAL INC. (US) 2007-04-17 US disclosed
WO-2005023804-A1 PEPTIDYL HETEROCYCLIC KETONE DERIVATIVES AND PREPARATION PROCESSES JANSSEN PHARMACEUTICA, N.V. (BE) 2005-03-17 WO disclosed