SCHEMBL8305799

SCHEMBL8305799

CC(C)OC(=O)N1CC[C@@](OCc2ccccc2)(c2ccc(Cl)cc2)[C@H](OCc2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.41
TACR1 P25103 3/20 0.39
OPRK1 P41145 2/20 0.38
OPRD1 P41143 1/20 0.38
TACR3 P29371 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6096715 0.89 CCR1 (0.40) CCR1TACR1TACR3
SCHEMBL6094587 0.89 CCR1 (0.40) CCR1TACR1TACR3
SCHEMBL6094255 0.89 CCR5 (0.40) CCR1TACR1OPRK1OPRD1
SCHEMBL6273383 0.89 CCR5 (0.40) CCR1TACR1OPRK1OPRD1
SCHEMBL6094257 0.89 CCR5 (0.40) CCR1TACR1OPRK1OPRD1
SCHEMBL8306441 0.89 CCR5 (0.40) CCR1TACR1OPRK1OPRD1
SCHEMBL6273386 0.89 CCR5 (0.40) CCR1TACR1OPRK1OPRD1
SCHEMBL6094878 0.88 OPRK1 (0.39) CCR1TACR1OPRK1OPRD1TACR3
SCHEMBL6094873 0.88 OPRK1 (0.39) CCR1TACR1OPRK1OPRD1TACR3
SCHEMBL8311127 0.81 DRD4 (0.41) TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080460-A1 SUBSTITUTED PIPERIDINES AS NOVEL MDM2-p53 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2004-09-23 WO disclosed