SCHEMBL8306010

SCHEMBL8306010

O=C(NCCCc1ccccc1)[C@H](Cc1ccccc1)NC(=O)[C@H]1N[C@@H]1C(=O)O.[Na]

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 2/20 0.50
KMT2A Q03164 3/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
CNR1 P21554 1/20 0.48
GRIA1 P42261 1/20 0.47
SRC P12931 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KDM4A O75164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7356782 0.94 GRIA1 (0.48) MMP8KMT2ACYP2D6CYP2C9CYP2C19
SCHEMBL7358942 0.91 KMT2A (0.53) MMP8KMT2AL3MBTL1
SCHEMBL7362788 0.89 MMP8 (0.48) MMP8KMT2ACYP2D6CYP2C9CYP2C19
SCHEMBL7363911 0.88 CHRNA1 (0.58) GRIA1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL7356539 0.87 L3MBTL1 (0.47) KMT2AGRIA1L3MBTL1CHRNB2CHRNB4
SCHEMBL8875868 0.86 PLG (0.53) KMT2AGRIA1L3MBTL1CHRNB2CHRNB4
SCHEMBL7356791 0.86 GRIA1 (0.47) MMP8KMT2ACYP2D6CYP2C9CYP2C19
SCHEMBL7362797 0.85 SRC (0.47) MMP8KMT2ACYP2D6CYP2C9CYP2C19
SCHEMBL7359233 0.85 BRS3 (0.51) KMT2ACNR1NPC1RAB9A
SCHEMBL7362904 0.84 LAP3 (0.51) KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0753003-B1 AZIRIDINE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-06-16 EP disclosed
US-5668128-A INHIBITORS OF THIOL PROTEASE, PROPHYLAXIS AND TREATMENT OF BONE DISEASES, OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-09-16 US disclosed