SCHEMBL8306016

SCHEMBL8306016

COC1(CC(=O)O)CCC(N2CCC(CCNc3ccncc3)CC2)CC1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTR2A P28223 1/20 0.35
HRH1 P35367 1/20 0.35
HTR2B P41595 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
ITGB3 P05106 4/20 0.34
ITGA2B P08514 4/20 0.34
CHRM4 P08173 5/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
ENPP1 P22413 1/20 0.33
RAB9A P51151 1/20 0.33
CCR2 P41597 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303583 0.86 KDM4E (0.40) GRIN2BCYP2D6CYP2C9KDM4EMEN1
SCHEMBL8300631 0.86 GRIN2B (0.40) GRIN2BCYP2D6CYP2C9HTR2AHRH1
SCHEMBL8301361 0.80 CYP2D6 (0.39) GRIN2BCYP2D6CYP2C9HTR2AHRH1
SCHEMBL8298652 0.79 ITGB3 (0.45) GRIN2BCYP2D6CYP2C9HTR2AHRH1
SCHEMBL8301158 0.75 CCR2 (0.35) GRIN2BCYP2D6CYP2C9HTR2AHRH1
SCHEMBL8614674 0.75 NAMPT (0.35) GRIN2BCYP2D6CYP2C9HRH3RAB9A
SCHEMBL8616373 0.74 CYP2D6 (0.32) GRIN2BCYP2D6CYP2C9ITGB3ITGA2B
SCHEMBL8304068 0.74 CYP2D6 (0.39) GRIN2BCYP2D6CYP2C9HTR2AHRH1
SCHEMBL8300686 0.72 NAMPT (0.43) GRIN2BCYP2D6CYP2C9HTR2AHRH1
SCHEMBL8300676 0.71 KDM4E (0.42) GRIN2BCYP2D6CYP2C9ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed
US-5786371-A INHIBIT AGGREGATION OF BLOOD PLATELETS BOEHRINGER MANNHEIM GMBH (DE) 1998-07-28 US disclosed