SCHEMBL8304068

SCHEMBL8304068

O=C(O)COCC1(O)CCC(N2CCC(CCCCNc3ccncc3)CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
GRIN2B Q13224 1/20 0.39
ITGB3 P05106 2/20 0.37
ITGA2B P08514 2/20 0.37
NAMPT P43490 10/20 0.36
GPR119 Q8TDV5 6/20 0.34
HTR2A P28223 1/20 0.33
HRH1 P35367 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301361 0.85 CYP2D6 (0.39) CYP2D6CYP2C9GRIN2BITGB3ITGA2B
SCHEMBL8306140 0.84 KDM4E (0.39) CYP2D6CYP2C9GRIN2BITGB3ITGA2B
SCHEMBL8300631 0.81 GRIN2B (0.40) CYP2D6CYP2C9GRIN2BITGB3ITGA2B
SCHEMBL8300686 0.80 NAMPT (0.43) CYP2D6CYP2C9GRIN2BITGB3ITGA2B
SCHEMBL8614674 0.79 NAMPT (0.35) CYP2D6CYP2C9GRIN2BNAMPTGPR119
SCHEMBL8303601 0.77 HRH3 (0.44) CYP2C9ITGB3ITGA2BHRH1
SCHEMBL8301126 0.74 KDM4E (0.40) CYP2D6CYP2C9GRIN2BHTR2A
SCHEMBL8306016 0.74 GRIN2B (0.38) CYP2D6CYP2C9GRIN2BITGB3ITGA2B
SCHEMBL8299936 0.73 KDM4E (0.41) CYP2D6
SCHEMBL8300039 0.72 ITGB3 (0.40) CYP2D6CYP2C9GRIN2BITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed