SCHEMBL8306253

SCHEMBL8306253

BrCc1conc1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 2/20 0.42
PTGS2 P35354 4/20 0.41
HSP90AA1 P07900 1/20 0.39
L3MBTL1 Q9Y468 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
NOTUM Q6P988 2/20 0.37
ERBB2 P04626 1/20 0.37
PTGS1 P23219 2/20 0.36
ALOX15 P16050 1/20 0.34
ALDH1A1 P00352 2/20 0.33
TRPA1 O75762 1/20 0.33
TSHR P16473 1/20 0.33
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28139688 0.81 NOTUM (0.44) GABRA5PTGS2HSP90AA1L3MBTL1TDP1
SCHEMBL23366325 0.81 PTGS2 (0.47) GABRA5PTGS2HSP90AA1L3MBTL1TDP1
SCHEMBL3213310 0.81 PTGS2 (0.41) GABRA5PTGS2HSP90AA1L3MBTL1TDP1
SCHEMBL2929388 0.81 NOTUM (0.49) GABRA5PTGS2HSP90AA1L3MBTL1TDP1
SCHEMBL5775916 0.78 NOTUM (0.46) GABRA5PTGS2HSP90AA1L3MBTL1TDP1
SCHEMBL5772931 0.78 PTGS2 (0.42) GABRA5PTGS2HSP90AA1L3MBTL1TDP1
SCHEMBL4973045 0.77 PTGS2 (0.41) GABRA5PTGS2HSP90AA1L3MBTL1TDP1
SCHEMBL27819710 0.77 KDM4E (0.49) GABRA5PTGS2HSP90AA1TDP1LMNA
SCHEMBL8168464 0.75 CYP19A1 (0.44) GABRA5PTGS2HSP90AA1PTGS1ALDH1A1
SCHEMBL11848234 0.74 PTGS2 (0.39) GABRA5PTGS2HSP90AA1L3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891339-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP disclosed
WO-1997036881-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO disclosed