SCHEMBL8306498

SCHEMBL8306498

CCN(c1ccncc1)c1csc2ncccc12

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
SLC6A2 P23975 4/20 0.34
PRKCI P41743 3/20 0.33
USP2 O75604 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
NPC1 O15118 1/20 0.31
HSP90AA1 P07900 1/20 0.31
HPGD P15428 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALOX15 P16050 1/20 0.30
RAB9A P51151 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8439568 0.89 POLB (0.45) ALDH1A1POLBKMT2ASLC6A2PRKCI
Hydrochloric Acid SCHEMBL8435449 0.88 POLB (0.44) ALDH1A1POLBKMT2ASLC6A2PRKCI
SCHEMBL8436327 0.87 KMT2A (0.38) ALDH1A1POLBKMT2ASLC6A2L3MBTL1
Hydrochloric Acid SCHEMBL8436071 0.86 KMT2A (0.38) ALDH1A1POLBKMT2ASLC6A2L3MBTL1
SCHEMBL8435363 0.81 CHKA (0.36) ALDH1A1KMT2ASLC6A2PRKCIL3MBTL1
SCHEMBL8056316 0.80 SLC6A2 (0.38) ALDH1A1SLC6A2HPGDMAPT
Hydrochloric Acid SCHEMBL8039091 0.79 ALDH1A1 (0.40) ALDH1A1SLC6A2HPGDMAPT
SCHEMBL8436069 0.78 TRPM8 (0.35) ALDH1A1SLC6A2USP2NPC1HPGD
SCHEMBL8439461 0.78 ALDH1A1 (0.34) ALDH1A1SLC6A2L3MBTL1NPC1HSP90AA1
SCHEMBL8439945 0.76 LMNA (0.34) ALDH1A1KMT2ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5252581-A Modulators of neurotransmitters HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-10-12 US claimed
WO-2004082686-A2 USE OF COMPOUNDS WITH COMBINED 5-HT1A AND SSRI ACTIVITIES TO TREAT SEXUAL DYSFUNCTION DYNOGEN PHARMACEUTICALS, INC. (US) 2004-09-30 WO disclosed
US-5856335-A GLYCINE PARTIAL AGONISTS. HOECHST MARION ROUSSEL, INC. (US) 1999-01-05 US disclosed
EP-0581106-B1 Substituted aminothienopyridines, a process for their preparation and their use as medicaments HOECHST MARION ROUSSEL INC (US) 1998-05-20 EP disclosed
US-5519032-A ANTIDEPRESSANTS, ANXIOLYTICS, ANTIEMETICS, ANTIPSYCHOTIC HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
EP-0581106-A1 Substituted aminothienopyridines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-02-02 EP disclosed
US-5252581-A Modulators of neurotransmitters HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-10-12 US disclosed