SCHEMBL8306791

SCHEMBL8306791

O=C(CCC(=O)N1CCC[C@H]1C(O)C(=O)O)NC1c2ccccc2-c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.46
TSHR P16473 2/20 0.42
SLC6A1 P30531 2/20 0.40
ACE P12821 8/20 0.38
ACE2 Q9BYF1 2/20 0.38
PREP P48147 1/20 0.38
FAP Q12884 1/20 0.38
F2 P00734 1/20 0.37
KMT2A Q03164 1/20 0.37
DUT P33316 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8994550 0.87 MAPT (0.40) MAPTTSHRACEACE2KMT2A
SCHEMBL7291931 0.81 MAPT (0.49) MAPTTSHRACEACE2F2
SCHEMBL7265245 0.80 MAPT (0.47) MAPTTSHRPREPFAPF2
SCHEMBL9873842 0.77 PREP (0.62) MAPTSLC6A1ACEACE2PREP
SCHEMBL9873839 0.77 PREP (0.62) MAPTSLC6A1ACEACE2PREP
SCHEMBL769700 0.74 MAPT (0.45) MAPTTSHRF2KMT2A
SCHEMBL8994595 0.73 F2 (0.43) MAPTTSHRACEACE2FAP
SCHEMBL8304030 0.73 ACE (0.36) SLC6A1ACEACE2PREPFAP
SCHEMBL7283530 0.73 MEN1 (0.51) SLC6A1ACEACE2KMT2A
SCHEMBL7290889 0.72 CHRM2 (0.43) SLC6A1ACEACE2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537802-B1 N-acylpyrrolidines, process for their preparation and their use for prevention and/or treatment of amnesia ONO PHARMACEUTICAL CO (JP) 1999-08-25 EP claimed
US-5545657-A 1-ALKYLOYLPYRROLIDIN-2-YLOXOALKANOIC ACIDS AND DERIVATIVES; ANTIAMNESIA AGENTS; INHIBITORS OF PROLYL ENDOPEPTIDASE; SUPPRESSION OF NEUROTRANSMITTER METABOLISM ONO PHARMACEUTICAL CO., LTD. (JP) 1996-08-13 US claimed
EP-0537802-A2 N-acylpyrrolidines and N-acylthiazolidines, process for their preparation and their use for prevention and/or treatment of amnesia ONO PHARMACEUTICAL CO., LTD. (JP) 1993-04-21 EP claimed