SCHEMBL8306794

SCHEMBL8306794

CC1(C)[C@]2(O)[C@@H](CO)O[C@@H](n3cnc4c(NCl)ncnc43)[C@]12O

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.49
ADORA2A P29274 6/20 0.48
ADORA1 P30542 5/20 0.48
ADORA2B P29275 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15633799 0.90 ADORA3 (0.50) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL5987749 0.86 ADORA2A (0.47) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL118827 0.85 ADORA3 (0.69) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL5786575 0.84 ADORA2A (0.48) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL121441 0.84 ADORA3 (0.69) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL1078828 0.84 ADORA2A (0.64) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL2294592 0.82 ADORA3 (0.43) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL122980 0.80 ADORA1 (0.72) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL6870926 0.79 ADORA3 (0.44) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL21480369 0.77 ADORA3 (0.58) ADORA3ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912520-A4 COMPOUNDS HAVING ANTIHYPERTENSIVE, CARDIOPROTECTIVE, ANTI-ISCHEMIC AND ANTILIPOLYTIC PROPERTIES RHONE POULENC RORER PHARMA (US) 1999-10-06 EP disclosed
EP-0912520-A1 COMPOUNDS HAVING ANTIHYPERTENSIVE, CARDIOPROTECTIVE, ANTI-ISCHEMIC AND ANTILIPOLYTIC PROPERTIES RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1999-05-06 EP disclosed
WO-1998001426-A1 COMPOUNDS HAVING ANTIHYPERTENSIVE, CARDIOPROTECTIVE, ANTI-ISCHEMIC AND ANTILIPOLYTIC PROPERTIES RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-01-15 WO disclosed