SCHEMBL8306927

SCHEMBL8306927

COC(=O)CC(N[C@H](C(N)=O)c1ccccc1)c1ccc(OC)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.50
GPR88 Q9GZN0 1/20 0.49
ATM Q13315 1/20 0.48
CNR2 P34972 2/20 0.47
DCAF1 Q9Y4B6 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
TNF P01375 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
PLA2G1B P04054 1/20 0.44
ATG4B Q9Y4P1 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CRHBP P24387 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44
CRHR2 Q13324 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303021 0.93 ALDH1A1 (0.47) EPHX1ATMDCAF1MEN1KMT2A
SCHEMBL8305547 0.85 CNR2 (0.45) CNR2MEN1KMT2ACYP1A2CYP3A4
SCHEMBL4854181 0.85 GPR88 (0.52) GPR88CNR2L3MBTL1MEN1KMT2A
SCHEMBL8306436 0.80 ALDH1A1 (0.47) EPHX1GPR88MEN1KMT2ACYP1A2
SCHEMBL4846798 0.79 TDP1 (0.53) GPR88ATMMEN1KMT2APLA2G1B
SCHEMBL4852606 0.79 PLA2G1B (0.55) GPR88ATMCNR2L3MBTL1MEN1
SCHEMBL8305705 0.79 EPHX1 (0.45) EPHX1CNR2DCAF1LMNACYP1A2
SCHEMBL1429119 0.79 KMT2A (0.60) GPR88CNR2L3MBTL1MEN1KMT2A
SCHEMBL3308208 0.79 ALDH1A1 (0.55) GPR88L3MBTL1MEN1KMT2ALMNA
SCHEMBL4561568 0.77 KDM4E (0.49) EPHX1GPR88MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed