SCHEMBL8305547

SCHEMBL8305547

COC(=O)CC(N[C@H](C(N)=O)c1ccccc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.45
EEF2K O00418 2/20 0.45
TACR1 P25103 2/20 0.43
CACNA1F O60840 1/20 0.43
CACNA1D Q01668 1/20 0.43
CACNA1S Q13698 1/20 0.43
CACNA1C Q13936 1/20 0.43
CACNA1A O00555 1/20 0.42
CACNA2D1 P54289 1/20 0.42
CACNB1 Q02641 1/20 0.42
LDHA P00338 1/20 0.41
LDHB P07195 1/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
FFAR1 O14842 1/20 0.41
SCN9A Q15858 1/20 0.40
PDPK1 O15530 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303021 0.89 ALDH1A1 (0.47) TACR1MEN1POLBKMT2AALDH1A1
SCHEMBL8306927 0.85 EPHX1 (0.50) CNR2MEN1KMT2ACYP1A2CYP3A4
SCHEMBL7994713 0.78 MEN1 (0.58) CNR2EEF2KLDHALDHBMEN1
SCHEMBL8306436 0.76 ALDH1A1 (0.47) MEN1KMT2ACYP1A2CYP2D6ALDH1A1
SCHEMBL8305705 0.75 EPHX1 (0.45) CNR2CYP1A2CYP2C19CYP2D6ALDH1A1
SCHEMBL5364020 0.75 THRB (0.45) CNR2EEF2KLDHALDHBMEN1
SCHEMBL5312465 0.74 MEN1 (0.51) MEN1POLBKMT2ACYP3A4ALDH1A1
SCHEMBL24036553 0.74 THRB (0.47) CNR2EEF2KLDHALDHBMEN1
SCHEMBL3738074 0.74 UTS2R (0.43) CNR2TACR1MEN1KMT2ACYP1A2
SCHEMBL3738078 0.74 UTS2R (0.43) CNR2TACR1MEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed