SCHEMBL8307056

SCHEMBL8307056

Cc1cc2c(cc1N1CCNC1=N)NCCO2

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.43
HSD17B10 Q99714 2/20 0.43
MAPT P10636 1/20 0.43
KDM4E B2RXH2 1/20 0.41
GLA P06280 1/20 0.41
HPGD P15428 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
ATM Q13315 1/20 0.41
BRD4 O60885 1/20 0.32
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308098 0.95 ALDH1A1 (0.43) ALDH1A1GAAHSD17B10MAPTKDM4E
SCHEMBL8303929 0.84 ALDH1A1 (0.37) ALDH1A1GAAHSD17B10MAPTKDM4E
SCHEMBL9530316 0.81 ALDH1A1 (0.36) ALDH1A1GAAHSD17B10MAPTKDM4E
SCHEMBL8304048 0.81 ALDH1A1 (0.37) ALDH1A1GAAHSD17B10MAPTKDM4E
SCHEMBL8305148 0.81 ALDH1A1 (0.38) ALDH1A1GAAHSD17B10MAPTKDM4E
SCHEMBL8302741 0.80 TP53 (0.46) ALDH1A1GAAMAPT
SCHEMBL8306232 0.79 ALDH1A1 (0.36) ALDH1A1GAAHSD17B10MAPTKDM4E
SCHEMBL8301746 0.79 ALDH1A1 (0.33) ALDH1A1GAAHSD17B10MAPTKDM4E
SCHEMBL8301972 0.76 ALDH1A1 (0.33) ALDH1A1GAAHSD17B10MAPTKDM4E
SCHEMBL8304203 0.75 ADRA2A (0.34) ALDH1A1GAAHSD17B10MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0548254-B1 6- OR 7-(IMIDAZOLIDIN-2-YLIDENEAMINO)-1,4-BENZOXAZINES AS ALPHA ADRENERGIC AGENTS ALLERGAN INC (US) 1999-06-02 EP disclosed
EP-0548254-A1 6- or 7- (2-IMINO-2-IMIDAZOLIDINE)-1,4-BENZOXAZINES AS ALPHA ADRENERGIC AGENTS ALLERGAN, INC. (US) 1993-06-30 EP disclosed
WO-1992004345-A1 6- or 7- (2-IMINO-2-IMIDAZOLIDINE)-1,4-BENZOXAZINES AS ALPHA ADRENERGIC AGENTS ALLERGAN, INC. (US) 1992-03-19 WO disclosed
US-5091528-A Antiglaucoma, antidiarrhea agents, diuretics, vasoconstrictors ALLERGAN, INC. (US) 1992-02-25 US disclosed