SCHEMBL8307517

SCHEMBL8307517

Cc1c(SCc2cccs2)ccnc1CSc1nc2ccccc2[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.55
NPC1 O15118 7/20 0.55
CYP1A2 P05177 2/20 0.55
CYP2D6 P10635 2/20 0.55
CYP2C9 P11712 2/20 0.55
CYP2C19 P33261 2/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2E1 P05181 1/20 0.46
CYP2C8 P10632 1/20 0.46
CYP2B6 P20813 1/20 0.46
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
NOS2 P35228 1/20 0.45
SMN1; SMN2 Q16637 5/20 0.44
HSD17B10 Q99714 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
NFKB1 P19838 2/20 0.44
NFKB2 Q00653 2/20 0.44
RELA Q04206 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304066 0.87 NOS3 (0.50) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9275547 0.84 RAB9A (0.66) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9874235 0.84 RAB9A (0.62) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL12195201 0.83 RAB9A (0.61) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8309290 0.83 RAB9A (0.54) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8008219 0.82 RAB9A (0.56) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9279666 0.82 RAB9A (0.58) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8914605 0.82 NPC1 (0.60) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8412992 0.82 NPC1 (0.60) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9278218 0.82 RAB9A (0.60) RAB9ANPC1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683776-B1 SUBSTITUTED HETEROARYLALKYLTHIOPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-07 EP disclosed
US-5587389-A Substituted heteroarylaklylthiopyridines for controlling helicobacter bacteria BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-12-24 US disclosed
WO-1994019346-A1 SUBSTITUTED HETEROARYLALKYLTHIOPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1994-09-01 WO disclosed