SCHEMBL8308067

SCHEMBL8308067

CNC(=O)c1cc(-c2ccccn2)nc2ccc(S(=O)(=O)N3CCC(C)CC3)cc12

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.78
HTT P42858 3/20 0.71
ALDH1A1 P00352 7/20 0.58
MAPT P10636 4/20 0.58
CNR1 P21554 1/20 0.58
RXFP1 Q9HBX9 3/20 0.57
LMNA P02545 5/20 0.56
THRB P10828 1/20 0.56
PKM P14618 2/20 0.56
POLB P06746 2/20 0.56
ATM Q13315 1/20 0.56
TSHR P16473 1/20 0.53
CYP2D6 P10635 1/20 0.53
HSD17B10 Q99714 2/20 0.52
MAPK1 P28482 2/20 0.52
MEN1 O00255 2/20 0.52
KDM4E B2RXH2 3/20 0.52
HPGD P15428 1/20 0.52
GRM4 Q14833 1/20 0.52
APOBEC3G Q9HC16 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311188 0.91 KMT2A (0.74) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8303840 0.86 KMT2A (0.80) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8308627 0.81 KMT2A (0.73) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8311182 0.79 RXFP1 (0.61) KMT2AHTTALDH1A1RXFP1LMNA
SCHEMBL8304199 0.79 ALDH1A1 (0.70) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8308787 0.78 ALDH1A1 (0.79) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8311184 0.78 RXFP1 (0.60) KMT2AHTTALDH1A1MAPTRXFP1
SCHEMBL8308784 0.77 KMT2A (0.67) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8310878 0.76 ALDH1A1 (0.66) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8311946 0.76 KDM4E (0.61) KMT2AHTTALDH1A1MAPTRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed