SCHEMBL8303840

SCHEMBL8303840

COC(CNC(=O)c1cc(-c2ccccn2)nc2ccc(S(=O)(=O)N3CCC(C)CC3)cc12)OC

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.80
HTT P42858 1/20 0.70
LMNA P02545 6/20 0.60
THRB P10828 1/20 0.60
RXFP1 Q9HBX9 4/20 0.58
CYP2D6 P10635 1/20 0.58
ALDH1A1 P00352 5/20 0.52
MAPT P10636 2/20 0.52
CNR1 P21554 1/20 0.52
MEN1 O00255 4/20 0.51
PKM P14618 2/20 0.50
POLB P06746 1/20 0.50
ATM Q13315 1/20 0.50
XBP1 P17861 1/20 0.48
KDM4E B2RXH2 3/20 0.47
HPGD P15428 2/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
TSHR P16473 1/20 0.47
HCRTR1 O43613 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304067 0.87 LMNA (0.78) KMT2AHTTLMNATHRBRXFP1
SCHEMBL8308067 0.86 KMT2A (0.78) KMT2AHTTLMNATHRBRXFP1
SCHEMBL8311188 0.84 KMT2A (0.74) KMT2AHTTLMNATHRBRXFP1
SCHEMBL8308627 0.80 KMT2A (0.73) KMT2AHTTLMNATHRBRXFP1
SCHEMBL8304199 0.77 ALDH1A1 (0.70) KMT2AHTTLMNARXFP1ALDH1A1
SCHEMBL8308784 0.76 KMT2A (0.67) KMT2AHTTLMNATHRBRXFP1
SCHEMBL8308787 0.76 ALDH1A1 (0.79) KMT2AHTTLMNARXFP1ALDH1A1
SCHEMBL8303898 0.74 ALDH1A1 (0.67) KMT2AHTTLMNARXFP1ALDH1A1
SCHEMBL8305649 0.74 HTT (0.61) KMT2AHTTLMNATHRBRXFP1
SCHEMBL8311946 0.73 KDM4E (0.61) KMT2AHTTLMNATHRBRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed