SCHEMBL8308110

SCHEMBL8308110

CC(=O)NC[C@H](NC(=O)CNCc1cccc2ccccc12)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.47
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
FNTA P49354 1/20 0.45
FNTB P49356 1/20 0.45
ANPEP P15144 1/20 0.44
TACR1 P25103 1/20 0.43
OPRD1 P41143 1/20 0.43
MAPT P10636 1/20 0.43
MME P08473 1/20 0.43
ACE P12821 1/20 0.43
CPA1 P15085 1/20 0.43
ACE2 Q9BYF1 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
PIN1 Q13526 1/20 0.42
NQO2 P16083 1/20 0.42
DNM1 Q05193 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8794402 0.94 FOLH1 (0.43) FOLH1KMT2AMEN1ALDH1A1L3MBTL1
SCHEMBL7749727 0.89 OPRK1 (0.48) KMT2AMEN1ALDH1A1L3MBTL1ANPEP
Trifluoroacetic Acid SCHEMBL8793852 0.85 OPRK1 (0.46) KMT2AMEN1ALDH1A1L3MBTL1ANPEP
SCHEMBL8439130 0.81 FNTA (0.63) FOLH1KMT2AMEN1ALDH1A1L3MBTL1
SCHEMBL7751346 0.81 FNTA (0.63) FOLH1KMT2AMEN1ALDH1A1L3MBTL1
SCHEMBL24130549 0.79 PIN1 (0.55) KMT2AMEN1ALDH1A1OPRD1MAPT
SCHEMBL7788436 0.78 FOLH1 (0.56) FOLH1KMT2AMEN1ALDH1A1L3MBTL1
SCHEMBL5999001 0.74 NQO2 (0.62) KMT2AMEN1ALDH1A1ANPEPMAPT
SCHEMBL8673871 0.73 MME (0.63) KMT2AMEN1TACR1MMEACE
SCHEMBL2761181 0.73 MME (0.63) KMT2AMEN1TACR1MMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0952842-A2 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 1999-11-03 EP claimed
WO-1997038664-A2 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1997-10-23 WO claimed