SCHEMBL8308408

SCHEMBL8308408

COCC1CN(c2ccc3nc(C4CCC(O)O4)sc3c2)C(=O)O1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 4/20 0.36
GRM5 P41594 3/20 0.36
MAOB P27338 4/20 0.36
MAOA P21397 3/20 0.35
F10 P00742 2/20 0.35
F2 P00734 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303658 0.85 GRM2 (0.37) GRM2GRM5MAOBMAOA
SCHEMBL8308585 0.85 GRM2 (0.37) GRM2GRM5MAOBMAOA
SCHEMBL8305638 0.80 MAOB (0.42) GRM2GRM5MAOBMAOA
SCHEMBL8305866 0.76 MAOB (0.38) GRM2GRM5MAOBMAOA
SCHEMBL8303567 0.76 GRM2 (0.35) GRM2GRM5MAOBMAOA
SCHEMBL8303566 0.76 GRM2 (0.35) GRM2GRM5MAOBMAOA
SCHEMBL3505520 0.75 GRM2 (0.39) GRM2GRM5MAOBF10
SCHEMBL8305067 0.74 GRM2 (0.39) GRM2GRM5MAOBF10
SCHEMBL8305251 0.74 MAOA (0.36) GRM2GRM5MAOBMAOAF10
SCHEMBL3503318 0.74 GRM2 (0.37) GRM2GRM5MAOBMAOAF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609441-B1 Oxazolidone derivatives as monoamine oxidase inhibitors EISAI CO LTD (JP) 1999-07-21 EP disclosed
US-5475014-A Monoamine oxidase inhibor; antidepressant EISAI CO., LTD. (JP) 1995-12-12 US disclosed
EP-0609441-A1 OXAZOLIDONE DERIVATIVE Eisai Co., Ltd. (JP) 1994-08-10 EP disclosed