SCHEMBL8308501

SCHEMBL8308501

CC(=NOCCOc1ccc(CC2SC(=O)N(C(c3ccccc3)(c3ccccc3)c3ccccc3)C2=O)cc1)c1ccc(N(C)S(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.45
L3MBTL1 Q9Y468 3/20 0.42
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
TDP1 Q9NUW8 2/20 0.35
NPC1 O15118 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ALDH1A1 P00352 3/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
NR1H2 P55055 1/20 0.33
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
POLB P06746 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308499 1.00 PPARG (0.45) PPARGL3MBTL1MEN1KMT2ATDP1
SCHEMBL8309646 0.90 PPARG (0.48) PPARGMEN1NPC1GAAMAPT
SCHEMBL8309649 0.90 PPARG (0.48) PPARGMEN1NPC1GAAMAPT
SCHEMBL8304791 0.86 PPARG (0.47) PPARGL3MBTL1MEN1KMT2ANPC1
SCHEMBL8387697 0.86 PPARG (0.47) PPARGL3MBTL1MEN1KMT2ANPC1
SCHEMBL8307062 0.86 PPARG (0.55) PPARGGAAMAPTHTT
SCHEMBL8307060 0.86 PPARG (0.55) PPARGGAAMAPTHTT
SCHEMBL8305087 0.86 PPARG (0.51) PPARGL3MBTL1MEN1KMT2AALDH1A1
SCHEMBL8305089 0.86 PPARG (0.51) PPARGL3MBTL1MEN1KMT2AALDH1A1
SCHEMBL8308451 0.84 PPARG (0.49) PPARGL3MBTL1NPC1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972959-A Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY, LIMITED (JP) 1999-10-26 US disclosed
EP-0708098-B1 Oxime derivatives, their preparation and their therapeutic use SANKYO CO (JP) 1999-03-03 EP disclosed
EP-0708098-A1 Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1996-04-24 EP disclosed