SCHEMBL8309601

SCHEMBL8309601

COC(=O)Cn1nc(-c2cccc(Cl)c2)cc1C

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.52
NPSR1 Q6W5P4 2/20 0.47
LMNA P02545 2/20 0.47
PTGS2 P35354 1/20 0.47
GAA P10253 2/20 0.47
KDM4E B2RXH2 2/20 0.47
TSHR P16473 4/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPK1 P28482 1/20 0.46
TP53 P04637 2/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 2/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311952 0.86 LMNA (0.51) MAPTLMNAPTGS2GAAKDM4E
SCHEMBL12122655 0.86 TSHR (0.60) MAPTLMNAKDM4ETSHRALDH1A1
SCHEMBL14982241 0.85 MAPT (0.56) MAPTNPSR1LMNAGAAKDM4E
SCHEMBL14982231 0.85 MAPT (0.50) MAPTNPSR1LMNAGAAKDM4E
SCHEMBL14982229 0.80 MAPT (0.44) MAPTGAAKDM4ETSHRALDH1A1
SCHEMBL24039001 0.77 KDM4E (0.49) MAPTGAAKDM4ETSHRALDH1A1
SCHEMBL8310550 0.76 PTGS2 (0.48) MAPTPTGS2GAAMAPK1
SCHEMBL1160614 0.76 TSHR (0.52) LMNAKDM4ETSHRALDH1A1MAPK1
SCHEMBL14982223 0.74 HTT (0.44) MAPTLMNAGAAKDM4ETSHR
SCHEMBL24638211 0.74 MAPT (0.38) MAPTLMNAGAAKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945437-A1 Pyrazolyl acrylic acid- and pyrazolyl oximino-acetic acid derivatives, their preparation and their use as fungicides SDS Biotech K.K. (JP) 1999-09-29 EP disclosed