SCHEMBL8309848

SCHEMBL8309848

O=[N+]([O-])c1ccc2ncnc(Nc3ccc(OCc4ccccn4)cc3F)c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
MAPT P10636 4/20 0.57
HTT P42858 4/20 0.57
EGFR P00533 7/20 0.53
L3MBTL1 Q9Y468 1/20 0.52
ALK Q9UM73 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
POLB P06746 2/20 0.47
NPC1 O15118 1/20 0.47
DUSP3 P51452 1/20 0.47
PTPN5 P54829 1/20 0.47
PTPN11 Q06124 1/20 0.47
GAA P10253 1/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
TNF P01375 1/20 0.45
CRHBP P24387 1/20 0.45
MAPK1 P28482 1/20 0.45
CRHR2 Q13324 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306485 0.85 EGFR (0.53) MAPTEGFRMEN1KMT2AERBB2
SCHEMBL8305114 0.84 EGFR (0.49) MAPTEGFRMEN1KMT2AERBB2
SCHEMBL8309481 0.82 EGFR (0.50) MAPTEGFRMEN1KMT2AERBB2
SCHEMBL8309434 0.81 EGFR (0.66) EGFRERBB2ERBB4CCNT1GSK3B
SCHEMBL8306919 0.81 KDR (0.65) EGFRERBB2ERBB4
SCHEMBL8620298 0.80 LMNA (0.41) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL3244620 0.79 EGFR (0.70) ALDH1A1MAPTHTTEGFRL3MBTL1
SCHEMBL8782984 0.79 DYRK1A (0.53) MAPTEGFRMEN1KMT2AERBB2
SCHEMBL8308072 0.79 EGFR (0.49) ALDH1A1EGFRERBB2ERBB4CCNT1
SCHEMBL8443996 0.78 CYP3A4 (0.54) MAPTEGFRMEN1KMT2AERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed