SCHEMBL8309981

SCHEMBL8309981

Nc1ccc(C(O)c2nccs2)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CYP3A4 P08684 3/20 0.35
TSHR P16473 3/20 0.35
ALOX5 P09917 1/20 0.34
CTSA P10619 5/20 0.34
RECQL P46063 2/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 2/20 0.33
HSD17B10 Q99714 2/20 0.33
FBP1 P09467 1/20 0.33
THRB P10828 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33
NOS1 P29475 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31090349 0.74 ALOX5 (0.41) TSHRALOX5CTSARECQLNPC1
SCHEMBL17064896 0.74 ALOX5 (0.53) CA1CA2ALOX5CTSAPRKDC
SCHEMBL8810387 0.73 ALOX5 (0.37) TSHRALOX5CTSANPC1RAB9A
SCHEMBL8308015 0.72 JAK2 (0.43) CA1CA2CYP3A4TSHRRECQL
SCHEMBL5655397 0.72 MAPT (0.44) CA1CA2CYP3A4TSHRRECQL
SCHEMBL8561583 0.71 CTSA (0.43) ALOX5CTSANPC1LMNARAB9A
SCHEMBL4768669 0.71 ALDH1A1 (0.42) TSHRALOX5CTSALMNAALDH1A1
SCHEMBL4849513 0.70 CTSA (0.48) CTSA
SCHEMBL6011470 0.68 FFAR2 (0.46) ALOX5CTSALMNASMN1; SMN2FBP1
SCHEMBL21788696 0.68 CA1 (0.42) CA1CA2CYP3A4TSHRRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed
US-5821246-A USEFUL AS TYROSINE KINASE INHIBITORS AND FOR THE TREATMENT OF PROLIFERATIVE DISEASES SUCH AS CANCER ZENECA LIMITED (GB) 1998-10-13 US disclosed
EP-0790986-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1997-08-27 EP disclosed
WO-1996015118-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1996-05-23 WO disclosed