SCHEMBL8310282

SCHEMBL8310282

Cc1oc2cc(N)cc(C)c2c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 1/20 0.35
DYRK1A Q13627 1/20 0.35
DYRK2 Q92630 1/20 0.35
ALDH1A1 P00352 7/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
CASP1 P29466 2/20 0.34
CASP7 P55210 2/20 0.34
CA9 Q16790 2/20 0.34
HSD17B10 Q99714 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
THRB P10828 1/20 0.34
ALDH2 P05091 4/20 0.33
ALDH1A2 O94788 3/20 0.33
ALDH1B1 P30837 3/20 0.33
TSHR P16473 2/20 0.33
ALDH1A3 P47895 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12925985 0.78 L3MBTL1 (0.49) ALDH1A1KDM4EHPGDTHRBALDH2
SCHEMBL8310517 0.72 CDK9 (0.36) CDK9DYRK1ADYRK2ALDH2ALDH1A2
SCHEMBL3234704 0.71 ADORA3 (0.43) CDK9DYRK1ADYRK2ALDH1A1KDM4E
SCHEMBL4958377 0.71 ALDH2 (0.38) ALDH1A1KDM4EHPGDCASP1CASP7
Hydrochloric Acid SCHEMBL8308661 0.71 CDK9 (0.35) CDK9DYRK1ADYRK2ALDH2ALDH1A2
SCHEMBL7082421 0.69 TPMT (0.41) ALDH1A1KDM4EHPGDCASP1CASP7
Hydrochloric Acid SCHEMBL7087423 0.68 TPMT (0.39) ALDH1A1KDM4EHPGDCASP1CASP7
SCHEMBL7086140 0.68 ALDH2 (0.41) ALDH1A1KDM4EHPGDCASP1CASP7
Oxalic Acid SCHEMBL8311094 0.67 KMT2A (0.33) ALDH1A1KDM4ETHRBALDH2ALDH1A2
SCHEMBL9205430 0.67 ELANE (0.37) ALDH1A1CA9CA1ALDH2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-A1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS Takeda Chemical Industries, Ltd. (JP) 1999-06-23 EP disclosed
WO-1998008842-A1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-05 WO disclosed