SCHEMBL8310409

SCHEMBL8310409

CC1(C)C=C(c2cccc[n+]2[O-])c2cc(Cl)ccc2OC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 2/20 0.39
ABCC8 Q09428 2/20 0.39
KCNJ11 Q14654 2/20 0.39
KCNJ8 Q15842 2/20 0.39
CYP19A1 P11511 1/20 0.33
MGAT2 Q10469 1/20 0.33
PGR P06401 1/20 0.33
AR P10275 1/20 0.33
MAOB P27338 1/20 0.32
ADRA2A P08913 3/20 0.32
DRD2 P14416 3/20 0.31
DRD4 P21917 3/20 0.31
CHRM2 P08172 2/20 0.31
HTR1A P08908 2/20 0.31
ADRA2B P18089 2/20 0.31
ADRA2C P18825 2/20 0.31
DRD1 P21728 2/20 0.31
SLC6A2 P23975 2/20 0.31
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314327 0.87 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8CYP19A1
SCHEMBL8310464 0.87 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8CYP19A1
SCHEMBL8312666 0.87 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8312815 0.86 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8CYP19A1
SCHEMBL8316384 0.85 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8KCNH2
SCHEMBL8311451 0.85 HTR2B (0.39) ABCC9ABCC8KCNJ11KCNJ8PGR
SCHEMBL8313863 0.84 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8ALDH1A1
SCHEMBL8315406 0.84 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8314966 0.84 KDM4E (0.39) ABCC9ABCC8KCNJ11KCNJ8CYP19A1
SCHEMBL8315805 0.84 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP claimed
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5652252-A POTASSIUM CHANNEL ACTIVATORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-07-29 US disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed