SCHEMBL8314966

SCHEMBL8314966

COc1ccc2c(c1)C(c1cccc[n+]1[O-])=CC(C)(C)CO2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
NPC1 O15118 1/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ABCC9 O60706 2/20 0.38
ABCC8 Q09428 2/20 0.38
KCNJ11 Q14654 2/20 0.38
KCNJ8 Q15842 2/20 0.38
CYP19A1 P11511 3/20 0.37
HTR2B P41595 2/20 0.37
SIGMAR1 Q99720 2/20 0.37
HTR7 P34969 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
PPIB P23284 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311836 0.87 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8DRD4
SCHEMBL8311394 0.85 ABCC9 (0.39) KDM4EALDH1A1MAPTNPC1HPGD
SCHEMBL8314327 0.85 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8CYP19A1
SCHEMBL8310464 0.85 ABCC9 (0.41) MAPTABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8310409 0.84 ABCC9 (0.39) ALDH1A1GAAMAPTSMN1; SMN2TDP1
SCHEMBL8312815 0.84 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8CYP19A1
SCHEMBL8316384 0.83 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8OPRD1
SCHEMBL8311451 0.83 HTR2B (0.39) ABCC9ABCC8KCNJ11KCNJ8HTR2B
SCHEMBL8315406 0.82 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8315805 0.82 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP claimed
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5652252-A POTASSIUM CHANNEL ACTIVATORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-07-29 US disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed