SCHEMBL8310504

SCHEMBL8310504

Cc1ccccc1S(=O)(=O)NC(=O)c1ccccc1COc1ccc2oc(-c3nc(C(C)(C)C)cs3)cc2c1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 12/20 0.43
RAPGEF3 O95398 1/20 0.38
SLC26A4 O43511 2/20 0.37
ALKBH2 Q6NS38 1/20 0.35
ALKBH3 Q96Q83 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
BCAT1 P54687 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311549 0.90 PTGER4 (0.40) PTGER4RAPGEF3SLC26A4
SCHEMBL8313568 0.87 CYSLTR2 (0.42) PTGER4RAPGEF3ALKBH2ALKBH3
SCHEMBL8310775 0.84 MAOB (0.42) SLC26A4KMT2A
SCHEMBL8316517 0.84 BCL2 (0.43) PTGER4SLC26A4MEN1KMT2A
SCHEMBL9400022 0.82 PTPRG (0.40) PTGER4ALKBH2ALKBH3MEN1KMT2A
SCHEMBL210686 0.79 PPARD (0.42) PTGER4SLC26A4MEN1KMT2A
SCHEMBL29623656 0.79 PPARD (0.42) PTGER4SLC26A4MEN1KMT2A
SCHEMBL8784066 0.79 PTGER4 (0.46) PTGER4RAPGEF3SLC26A4MEN1KMT2A
Hydrochloric Acid SCHEMBL1224090 0.78 PPARD (0.41) PTGER4SLC26A4MEN1KMT2A
SCHEMBL6598204 0.78 ALKBH2 (0.39) PTGER4ALKBH2ALKBH3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528337-B1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-10-20 EP disclosed
US-5296495-A Antiallergens, antiinflammatory FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US disclosed
EP-0528337-A1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-02-24 EP disclosed