SCHEMBL8311161

SCHEMBL8311161

CC(=O)Nc1cccn2c(C(C)=NO)c(C)nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
LMNA P02545 1/20 0.43
GLA P06280 1/20 0.43
ALDH1A1 P00352 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
KMT2A Q03164 3/20 0.40
HPGD P15428 1/20 0.40
KDM4E B2RXH2 2/20 0.36
GAA P10253 1/20 0.36
GUCY1B2 O75343 1/20 0.36
GUCY1A2 P33402 1/20 0.36
GUCY1A1 Q02108 1/20 0.36
GUCY1B1 Q02153 1/20 0.36
TP53 P04637 3/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
HCRTR1 O43613 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312406 1.00 CYP1A2 (0.46) CYP1A2LMNAGLAALDH1A1SMN1; SMN2
SCHEMBL8317131 0.79 ALDH1A1 (0.46) LMNAGLAALDH1A1SMN1; SMN2KMT2A
SCHEMBL9281511 0.75 CYP1A2 (0.50) CYP1A2LMNAGLAALDH1A1SMN1; SMN2
SCHEMBL8311289 0.71 SMN1; SMN2 (0.59) ALDH1A1SMN1; SMN2KMT2AKDM4ETP53
SCHEMBL9080957 0.70 KMT2A (0.46) ALDH1A1SMN1; SMN2KMT2AHPGDMAPT
SCHEMBL8312072 0.70 KMT2A (0.67) LMNAGLAALDH1A1SMN1; SMN2KMT2A
SCHEMBL3551654 0.68 ALDH1A1 (0.67) CYP1A2GLAALDH1A1SMN1; SMN2KMT2A
SCHEMBL9230500 0.68 EPHB3 (0.46) ALDH1A1SMN1; SMN2KMT2AHPGDMAPT
SCHEMBL28549246 0.66 ALDH1A1 (0.63) CYP1A2GLAALDH1A1SMN1; SMN2KMT2A
SCHEMBL7989395 0.66 KMT2A (0.56) CYP1A2ALDH1A1SMN1; SMN2KMT2AGUCY1B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0649425-B1 PYRIDINO-, PYRROLIDINO- AND AZEPINO-SUBSTITUTED OXIMES USEFUL AS ANTI-ATHEROSCLEROSIS AND ANTI-HYPERCHOLESTEROLEMIC AGENTS UPJOHN CO (US) 1999-03-10 EP claimed