SCHEMBL8311491

SCHEMBL8311491

CCc1cc(NC)ccc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
SLC18A1 P54219 1/20 0.37
SLC18A2 Q05940 1/20 0.37
HPGD P15428 1/20 0.37
PLA2G1B P04054 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
ATG4B Q9Y4P1 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34
KCNH2 Q12809 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14270576 0.84 TAAR1 (0.36) TSHRSLC18A1SLC18A2PLA2G1BCYP1A2
SCHEMBL16838138 0.83 CYP1A2 (0.35) TSHRSLC18A1SLC18A2HPGDPLA2G1B
SCHEMBL15250773 0.83 SLC18A1 (0.37) TSHRSLC18A1SLC18A2HPGDKMT2A
SCHEMBL27680833 0.82 SLC18A1 (0.40) TSHRSLC18A1SLC18A2HPGDPLA2G1B
SCHEMBL16838137 0.82 MAPK1 (0.37) TSHRSLC18A1SLC18A2PLA2G1BCYP1A2
SCHEMBL15030165 0.80 ALDH1A1 (0.42) PLA2G1BCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL19290592 0.79 ALDH1A1 (0.38) TSHRHPGDPLA2G1BCYP1A2CYP3A4
SCHEMBL16715358 0.77 ADRA2C (0.55) HPGDCYP2C9SMN1; SMN2KCNH2ALDH1A1
SCHEMBL19232759 0.77 TSHR (0.35) TSHRHPGDPLA2G1BCYP1A2CYP3A4
SCHEMBL6724337 0.77 TSHR (0.45) TSHRHPGDSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3919474-B1 HBV INHIBITOR AND USE THEREOF XIAN XINTONG PHARMACEUTICAL RES CO LTD (CN) 2023-10-11 EP disclosed
EP-1944305-B1 Quinoline derivatives as phosphodiesterase inhibitors GLAXO GROUP LTD (GB) 2011-10-19 EP disclosed
CN-101815710-A Pyrimidine and pyridine derivatives, their pharmaceutical use and compositions PFIZER 2010-08-25 CN disclosed
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP disclosed
WO-2004103998-A1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LIMITED (GB) 2004-12-02 WO disclosed