SCHEMBL8312456

SCHEMBL8312456

COC(=O)/C=C/c1cc2c(s1)CCNC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 4/20 0.51
TPSAB1 Q15661 1/20 0.40
TPSD1 Q9BZJ3 1/20 0.40
TPSG1 Q9NRR2 1/20 0.40
ITGB3 P05106 5/20 0.38
ITGA2B P08514 5/20 0.38
TTR P02766 1/20 0.38
APP P05067 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
TYR P14679 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
PARP1 P09874 3/20 0.36
PARP2 Q9UGN5 3/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
PTPN1 P18031 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4760446 0.83 PNMT (0.52) PNMTTPSAB1TPSD1TPSG1ITGB3
SCHEMBL4760447 0.83 PNMT (0.52) PNMTTPSAB1TPSD1TPSG1ITGB3
SCHEMBL5648139 0.82 PNMT (0.46) PNMTTPSAB1TPSD1TPSG1ITGB3
Trifluoroacetic Acid SCHEMBL5648133 0.77 PNMT (0.46) PNMTTPSAB1TPSD1TPSG1ITGB3
Trifluoroacetic Acid SCHEMBL5648145 0.77 PNMT (0.46) PNMTTPSAB1TPSD1TPSG1ITGB3
SCHEMBL2559315 0.74 PNMT (0.56) PNMTTPSAB1TPSD1TPSG1ITGB3
SCHEMBL977061 0.73 PNMT (0.70) PNMTTPSAB1TPSD1TPSG1ITGB3
SCHEMBL3175428 0.73 TTR (0.52) PNMTTTRAPPCA12CA1
SCHEMBL3175417 0.73 TTR (0.52) PNMTTTRAPPCA12CA1
Hydrochloric Acid SCHEMBL6421343 0.72 PNMT (0.68) PNMTTPSAB1TPSD1TPSG1ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7265128-B2 3-amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes MERCK & CO., INC. (US) 2007-09-04 US disclosed
US-7265128-B2 3-amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes MERCK & CO., INC. (US) 2007-09-04 US disclosed
WO-2004064778-A2 3-AMINO-4-PHENYLBUTANOIC ACID DERIVATIVES AS DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES MERCK & CO. INC. (US) 2004-08-05 WO disclosed