SCHEMBL8313290

SCHEMBL8313290

Clc1cccc(C(=C2CCNCC2)c2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 9/20 0.49
OPRD1 P41143 9/20 0.49
OPRK1 P41145 4/20 0.49
KCNH2 Q12809 2/20 0.45
ABCB11 O95342 1/20 0.45
HTR2A P28223 3/20 0.41
HTR2B P41595 3/20 0.41
CYP2D6 P10635 2/20 0.41
HTR3A P46098 2/20 0.41
SETD7 Q8WTS6 1/20 0.41
LMNA P02545 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
HRH1 P35367 1/20 0.41
CHRNA4 P43681 1/20 0.41
HTR2C P28335 4/20 0.40
PARP1 P09874 1/20 0.40
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315518 0.95 OPRM1 (0.46) OPRM1OPRD1OPRK1KCNH2ABCB11
SCHEMBL8314573 0.85 OPRD1 (0.58) OPRM1OPRD1OPRK1KCNH2ABCB11
SCHEMBL2457390 0.84 OPRD1 (0.61) OPRM1OPRD1OPRK1KCNH2ABCB11
Bromide SCHEMBL10598951 0.82 OPRD1 (0.59) OPRM1OPRD1OPRK1KCNH2ABCB11
Hydrochloric Acid SCHEMBL7647391 0.82 OPRD1 (0.59) OPRM1OPRD1OPRK1KCNH2ABCB11
SCHEMBL13437760 0.80 OPRM1 (0.56) OPRM1OPRD1OPRK1LMNATP53
SCHEMBL10461671 0.77 OPRM1 (0.67) OPRM1OPRD1OPRK1KCNH2ABCB11
SCHEMBL10460871 0.77 OPRD1 (0.65) OPRM1OPRD1OPRK1KCNH2ABCB11
SCHEMBL9434960 0.76 OPRD1 (0.57) OPRM1OPRD1OPRK1KCNH2ABCB11
SCHEMBL22491524 0.75 OPRM1 (0.50) OPRM1OPRD1OPRK1KCNH2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536419-B1 TRICYCLIC TRIAZOLE DERIVATIVES, PRODUCTION AND USE THEREOF TORAY INDUSTRIES (JP) 1999-10-13 EP disclosed
CN-1033327-C Process for preparing tricyclotriazolo derivatives and their use TORAY INDUSTRIES (JP) 1996-11-20 CN disclosed
EP-0536419-A1 TRICYCLIC TRIAZOLE DERIVATIVE, PRODUCTION THEREOF, AND USE THEREOF TORAY INDUSTRIES, INC. (JP) 1993-04-14 EP disclosed
CN-1066849-A Three ring triazolo derivatives, its Manufacturing approach and use TORAY INDUSTRIES (JP) 1992-12-09 CN disclosed