SCHEMBL8315518

SCHEMBL8315518

Clc1cccc(C(=C2CCNCC2)c2cccc(Cl)c2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 9/20 0.46
OPRD1 P41143 9/20 0.46
ABCB11 O95342 1/20 0.45
KCNH2 Q12809 1/20 0.45
OPRK1 P41145 4/20 0.44
HTR2C P28335 4/20 0.43
HTR2A P28223 2/20 0.43
HTR2B P41595 2/20 0.43
PARP1 P09874 1/20 0.43
HTR7 P34969 3/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
ADRB1 P08588 1/20 0.42
CYP3A4 P08684 1/20 0.42
HTR1A P08908 1/20 0.42
CYP2D6 P10635 1/20 0.42
THRB P10828 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313290 0.95 OPRM1 (0.49) OPRM1OPRD1ABCB11KCNH2OPRK1
SCHEMBL13437760 0.81 OPRM1 (0.56) OPRM1OPRD1OPRK1TP53THRB
SCHEMBL8314573 0.79 OPRD1 (0.58) OPRM1OPRD1ABCB11KCNH2OPRK1
SCHEMBL8316059 0.79 OPRM1 (0.49) OPRM1OPRD1ABCB11KCNH2OPRK1
SCHEMBL14415620 0.79 OPRD1 (0.65) OPRM1OPRD1ABCB11KCNH2OPRK1
Hydrochloric Acid SCHEMBL30055362 0.78 HTR2C (0.39) OPRM1OPRD1OPRK1HTR2CHTR2A
Hydrochloric Acid SCHEMBL27166047 0.78 HTR2C (0.39) OPRM1OPRD1OPRK1HTR2CHTR2A
SCHEMBL10460871 0.77 OPRD1 (0.65) OPRM1OPRD1ABCB11KCNH2OPRK1
SCHEMBL2457390 0.77 OPRD1 (0.61) OPRM1OPRD1ABCB11KCNH2OPRK1
Bromide SCHEMBL10598951 0.75 OPRD1 (0.59) OPRM1OPRD1ABCB11KCNH2OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536419-B1 TRICYCLIC TRIAZOLE DERIVATIVES, PRODUCTION AND USE THEREOF TORAY INDUSTRIES (JP) 1999-10-13 EP disclosed
US-5683998-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS, ANTIPAF AGENTS TORAY INDUSTRIES, INC. (JP) 1997-11-04 US disclosed
EP-0536419-A1 TRICYCLIC TRIAZOLE DERIVATIVE, PRODUCTION THEREOF, AND USE THEREOF TORAY INDUSTRIES, INC. (JP) 1993-04-14 EP disclosed