SCHEMBL8313716

SCHEMBL8313716

Oc1ccc2nc(CN3CCC(C(O)c4ccccc4)CC3)[nH]c2c1

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 9/20 0.67
GRIN2B Q13224 9/20 0.67
GAA P10253 2/20 0.49
TSHR P16473 2/20 0.49
PKM P14618 1/20 0.49
NPC1 O15118 1/20 0.48
KDM4E B2RXH2 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
DRD4 P21917 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5238060 0.92 GRIN1 (0.56) GRIN1GRIN2BGAATSHRNPC1
SCHEMBL8313723 0.81 GRIN1 (1.00) GRIN1GRIN2BGAATSHRPKM
SCHEMBL8312793 0.79 GRIN1 (0.67) GRIN1GRIN2BGAATSHRPKM
SCHEMBL8318192 0.75 GRIN1 (1.00) GRIN1GRIN2BGAANPC1DRD4
SCHEMBL8319076 0.74 GRIN1 (1.00) GRIN1GRIN2BGAANPC1DRD4
SCHEMBL7536655 0.73 KDM4E (0.61) TSHRKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8321110 0.73 GRIN1 (0.66) GRIN1GRIN2BGAATSHRPKM
SCHEMBL8318042 0.72 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8313704 0.72 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8320273 0.72 GRIN1 (1.00) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048364-A1 2-[(4-BENZYL)-1-PIPERIDINYL)METHYL]BENZIMIDAZOLE-5-OL DERIVATIVES AS NR2B RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2004-06-10 WO disclosed