SCHEMBL8313722

SCHEMBL8313722

O=C(c1ccccc1)C1CCN(CCCCl)CC1

nearest known ligand 0.71

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.71
HTR2A P28223 2/20 0.68
KDM4E B2RXH2 1/20 0.60
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
HRH3 Q9Y5N1 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20577435 0.91 HTR2A (0.71) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL11519875 0.87 KCNH2 (0.62) KCNH2HTR2AHRH3
SCHEMBL7250766 0.87 KCNH2 (0.72) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL9726195 0.86 HTR2A (0.69) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL11521416 0.86 MGLL (0.54) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL29448592 0.86 KCNH2 (0.69) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL11749648 0.84 HSD11B1 (0.54) KCNH2HTR2AKDM4ECYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9650868 0.83 HTR2A (0.82) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL7368435 0.83 HTR2A (0.83) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL24135454 0.82 KCNH2 (0.79) KCNH2HTR2AKDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536419-B1 TRICYCLIC TRIAZOLE DERIVATIVES, PRODUCTION AND USE THEREOF TORAY INDUSTRIES (JP) 1999-10-13 EP disclosed
US-5683998-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS, ANTIPAF AGENTS TORAY INDUSTRIES, INC. (JP) 1997-11-04 US disclosed
CN-1033327-C Process for preparing tricyclotriazolo derivatives and their use TORAY INDUSTRIES (JP) 1996-11-20 CN disclosed
EP-0536419-A1 TRICYCLIC TRIAZOLE DERIVATIVE, PRODUCTION THEREOF, AND USE THEREOF TORAY INDUSTRIES, INC. (JP) 1993-04-14 EP disclosed
CN-1066849-A Three ring triazolo derivatives, its Manufacturing approach and use TORAY INDUSTRIES (JP) 1992-12-09 CN disclosed
US-4151285-A ANTICONVULSANT, ANTI-ANXIETY AGENTS A. H. ROBINS COMPANY, INC. (US) 1979-04-24 US disclosed