SCHEMBL8313734

SCHEMBL8313734

CC1(C)C=C(c2ccccn2)c2ccc(Cl)c(Cl)c2OC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.36
NPC1 O15118 3/20 0.34
MAPT P10636 3/20 0.34
RAB9A P51151 3/20 0.34
PKM P14618 2/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KLF5 Q13887 1/20 0.33
CCR1 P32246 2/20 0.32
CCR5 P51681 2/20 0.32
CCR8 P51685 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
METAP1 P53582 1/20 0.32
BLM P54132 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313795 0.83 CCR1 (0.38) GRM5NPC1MAPTRAB9APKM
SCHEMBL8316296 0.81 CCR1 (0.35) GRM5NPC1MAPTRAB9APKM
SCHEMBL8316184 0.79 KDM4E (0.37) NPC1MAPTRAB9APKMTP53
SCHEMBL8312863 0.78 MAPT (0.39) GRM5NPC1MAPTRAB9APKM
SCHEMBL8315666 0.77 NTRK1 (0.35) GRM5NPC1MAPTRAB9APKM
SCHEMBL8315309 0.75 ADRA1A (0.38) GRM5NPC1MAPTRAB9APKM
SCHEMBL8313085 0.75 CCR1 (0.40) GRM5NPC1MAPTRAB9APKM
SCHEMBL8311427 0.73 SCN9A (0.35) GRM5RAB9AMAPK1ALDH1A1CCR1
SCHEMBL8315585 0.72 ADRA1A (0.40) GRM5NPC1MAPTRAB9APKM
SCHEMBL8314584 0.72 FABP6 (0.37) GRM5MAPTRAB9AMETAP1NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed