SCHEMBL8315666

SCHEMBL8315666

CC1(C)C=C(c2ccccn2)c2cc(F)c(Cl)cc2OC1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 8/20 0.35
NPC1 O15118 2/20 0.32
MAPT P10636 2/20 0.32
PKM P14618 2/20 0.32
RAB9A P51151 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
BACE1 P56817 1/20 0.32
KCNH2 Q12809 1/20 0.32
GRM5 P41594 3/20 0.32
KLF5 Q13887 1/20 0.31
FFAR1 O14842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311427 0.90 SCN9A (0.35) NTRK1RAB9AALDH1A1CCR1CCR5
SCHEMBL8316296 0.90 CCR1 (0.35) NTRK1NPC1MAPTPKMRAB9A
SCHEMBL8312863 0.82 MAPT (0.39) NPC1MAPTPKMRAB9AALDH1A1
SCHEMBL8314584 0.82 FABP6 (0.37) MAPTRAB9ABACE1GRM5
SCHEMBL8875966 0.79 NPY5R (0.34) CCR1CCR5CCR8
SCHEMBL8316488 0.79 PDE10A (0.40) NPC1MAPTPKMRAB9AALDH1A1
SCHEMBL8316184 0.79 KDM4E (0.37) NPC1MAPTPKMRAB9AALDH1A1
SCHEMBL8315486 0.78 NPC1 (0.39) NPC1MAPTPKMRAB9AALDH1A1
SCHEMBL8313795 0.78 CCR1 (0.38) NTRK1NPC1MAPTPKMRAB9A
SCHEMBL8315309 0.77 ADRA1A (0.38) NPC1MAPTPKMRAB9ACCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed