SCHEMBL8314569

SCHEMBL8314569

FC(F)(F)c1csc(-c2cc3cc(OCc4ccccc4CCl)ccc3o2)n1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.36
F2RL3 Q96RI0 3/20 0.35
PPARD Q03181 3/20 0.34
PPARA Q07869 1/20 0.34
CYP19A1 P11511 1/20 0.33
SLC26A4 O43511 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
PTGER4 P35408 1/20 0.32
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
TP53 P04637 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
S1PR1 P21453 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314208 0.90 F2RL3 (0.36) F2RL3CYP19A1SLC26A4MEN1KMT2A
SCHEMBL8310491 0.88 F2RL3 (0.33) ARF2RL3PPARDPPARACYP19A1
SCHEMBL8310753 0.85 ALDH1A1 (0.45) F2RL3CYP19A1SLC26A4MEN1KMT2A
SCHEMBL8315191 0.83 MAPK1 (0.41) F2RL3PPARDPPARACYP19A1MEN1
SCHEMBL8310707 0.83 F2RL3 (0.31) ARF2RL3PPARDPPARA
SCHEMBL8310437 0.83 F2RL3 (0.35) F2RL3CYP19A1SLC26A4MEN1KMT2A
SCHEMBL8316136 0.82 F2RL3 (0.36) F2RL3CYP19A1SLC26A4MEN1KMT2A
SCHEMBL8315476 0.82 CYP19A1 (0.43) F2RL3CYP19A1MEN1KMT2ATP53
SCHEMBL8314511 0.82 FFAR4 (0.39) F2RL3CYP19A1SLC26A4MEN1KMT2A
SCHEMBL8310727 0.81 MAPT (0.44) F2RL3CYP19A1MEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528337-B1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-10-20 EP disclosed
US-5296495-A Antiallergens, antiinflammatory FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-03-22 US disclosed
EP-0528337-A1 New thiazolylbenzofuran derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-02-24 EP disclosed