SCHEMBL8314686

SCHEMBL8314686

Cc1ccc(C)c(C(=O)Nc2ccc(C(=O)O)cc2Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.57
PPARG P37231 1/20 0.55
PPARA Q07869 1/20 0.55
NPC1 O15118 3/20 0.54
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 2/20 0.53
TAS1R3 Q7RTX0 2/20 0.52
TAS1R1 Q7RTX1 2/20 0.52
TAS1R2 Q8TE23 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.51
PYGL P06737 3/20 0.51
TP53 P04637 1/20 0.50
MEN1 O00255 1/20 0.50
GFER P55789 1/20 0.50
KMT2A Q03164 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
PDK1 Q15118 1/20 0.49
PDK2 Q15119 1/20 0.49
PDK3 Q15120 1/20 0.49
PDK4 Q16654 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17498480 0.88 RAB9A (0.56) RAB9APPARGPPARANPC1ALDH1A1
SCHEMBL7340569 0.87 PYGL (0.61) RAB9ANPC1KDM4EALDH1A1PYGL
SCHEMBL7332090 0.85 PYGL (0.62) RAB9APPARGNPC1KDM4EALDH1A1
SCHEMBL16160866 0.84 RAB9A (0.51) RAB9APPARGPPARANPC1ALDH1A1
SCHEMBL8812458 0.84 RAB9A (0.57) RAB9APPARGPPARANPC1KDM4E
SCHEMBL27561744 0.83 NR1H4 (0.57) PPARGPPARANPC1KDM4EALDH1A1
SCHEMBL6972628 0.82 RAB9A (0.58) RAB9APPARGPPARANPC1TAS1R3
SCHEMBL8313578 0.80 PYGL (0.56) RAB9APPARGNPC1KDM4EALDH1A1
SCHEMBL7372458 0.79 RAB9A (0.57) RAB9APPARGNPC1KDM4EALDH1A1
SCHEMBL6968515 0.78 PYGL (0.57) RAB9APPARGNPC1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636625-B1 Tricyclic diazepines vasopressin and oxytocin antagonists AMERICAN CYANAMID CO (US) 1999-01-27 EP disclosed