SCHEMBL6968515

SCHEMBL6968515

Cc1ccccc1-c1ccccc1C(=O)Nc1ccc(C(=O)O)cc1Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 2/20 0.57
RAB9A P51151 3/20 0.53
PPARG P37231 2/20 0.49
NR1H4 Q96RI1 1/20 0.49
GRM4 Q14833 1/20 0.49
TP53 P04637 1/20 0.49
GAA P10253 1/20 0.49
GRM1 Q13255 1/20 0.48
ALDH1A1 P00352 5/20 0.48
KDM4E B2RXH2 2/20 0.47
FTO Q9C0B1 1/20 0.47
PTGFR P43088 1/20 0.47
NPC1 O15118 2/20 0.46
MEN1 O00255 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
KCNH2 Q12809 1/20 0.46
PDK1 Q15118 1/20 0.46
PDK2 Q15119 1/20 0.46
PDK3 Q15120 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972628 0.91 RAB9A (0.58) PYGLRAB9APPARGNR1H4TP53
SCHEMBL7332090 0.90 PYGL (0.62) PYGLRAB9APPARGNR1H4GRM4
SCHEMBL7372458 0.85 RAB9A (0.57) PYGLRAB9APPARGNR1H4GAA
SCHEMBL6961250 0.85 ALDH1A1 (0.54) RAB9AGRM4TP53GAAALDH1A1
SCHEMBL8313578 0.85 PYGL (0.56) PYGLRAB9APPARGNR1H4GRM4
SCHEMBL27376893 0.82 PYGL (0.54) PYGLRAB9APPARGNR1H4ALDH1A1
SCHEMBL6968458 0.81 HCAR3 (0.66) RAB9AALDH1A1PTGFRNPC1MEN1
SCHEMBL8961733 0.81 HCAR3 (0.66) RAB9AALDH1A1PTGFRNPC1MEN1
SCHEMBL7331410 0.79 GRM4 (0.59) PYGLRAB9AGRM4TP53ALDH1A1
SCHEMBL8812458 0.78 RAB9A (0.57) PYGLRAB9APPARGTP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620216-B1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2003-01-08 EP disclosed
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed