SCHEMBL8314779

SCHEMBL8314779

CS(=O)(=O)c1ncc2ncnc(Nc3ccc(N)c(C#N)c3)c2n1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.45
CTSD P07339 2/20 0.39
BACE1 P56817 2/20 0.39
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
CCNA1 P78396 1/20 0.39
PIP4K2A P48426 1/20 0.39
BACE2 Q9Y5Z0 1/20 0.38
BRAF P15056 1/20 0.37
ERBB2 P04626 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318294 0.82 EGFR (0.46) EGFRCTSDBACE1BACE2
SCHEMBL6994593 0.82 ABCG2 (0.54) EGFR
SCHEMBL8319085 0.82 EGFR (0.44) EGFR
SCHEMBL6997375 0.79 EGFR (0.47) EGFRBRAFERBB2HPGDHTT
SCHEMBL8317145 0.79 EGFR (0.49) EGFRERBB2HPGDHTT
SCHEMBL8484295 0.78 EGFR (0.53) EGFRERBB2
SCHEMBL6417047 0.77 EGFR (0.66) EGFRERBB2HTT
SCHEMBL6993872 0.77 EGFR (0.69) EGFRHTT
SCHEMBL6992072 0.77 EGFR (0.44) EGFRBRAFERBB2HPGDHTT
SCHEMBL8486684 0.77 EGFR (0.46) EGFRBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed